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1-(4-Methoxyphenyl) -7-oxo-6-[4-(2-oxopiperidin-1-yl) phenyl] -4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine -3-carboxylic acid ethyl ester ikemikari yakaoma yemakemikari yakaratidza kukwanisa munzvimbo dzakasiyana-siyana dzemakemikari emishonga uye kuwanikwa kwezvinodhaka.Heino tsanangudzo yekushandiswa kwayo mumashoko anenge 300. Ichi chikwata, chinowanzonzi se ethyl ester derivative ye 1- (4-Methoxyphenyl) -7-oxo-6-[4- (2-oxopiperidin-1-yl) phenyl] -4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylic acid, ndeyekirasi yepyrazolo [3,4-c] pyridine derivatives.Zvigadzirwa izvi zvakakwezva kutarisa mukuwanikwa kwezvinodhaka nekuda kwekugona kwavo munzvimbo dzakasiyana-siyana dzokurapa.Kumwe kushandiswa kwekomboni iyi kunowanikwa mumunda wekurwisa kenza.Pyrazolo [3,4-c] pyridine derivatives yakaratidza inovimbisa anti-proliferative chiitiko kurwisa akati wandei ekenza maseru.Kugona kwavo kuvharidzira nzira dzakanangana mukukura kwebundu uye kurarama zvinovaita vanogona kukwikwidza mukugadzirwa kwemishonga inorwisa cancer.Zvimwe zvidzidzo zvinodiwa kuti uongorore maitiro echiito uye kuongorora kushanda kwekomboni mu preclinical uye kliniki zvirongwa.Uyezve, ichi chikamu chakaratidza chivimbiso sechinhu chinogona antibacterial agent.Yakaratidza chiitiko chinopesana nemhando dzakasiyana dzebhakitiriya, kusanganisira ese maGram-positive uye Gram-negative mabhakitiriya.Iko kugona kunongedza akawanda strains kunoratidza kugona kwayo mukurwisa mabhakitiriya asingaurayiwi nemishonga, ayo ave kukosha kwehutano hwepasirese.Kuwedzera kutsvakurudza kunobvumirwa kuongorora maitiro ayo uye kuongorora kushanda kwayo mukurwisana nehutachiona hwehutachiona.Kuwedzera, pyrazolo [3,4-c] pyridine derivatives, kusanganisira iyi komputa, yakaratidza kukwanisa mukurapa kwezvirwere zvinoputika uye autoimmune.Kuzvimba kunoita basa rakakosha mumamiriro akasiyana senge rheumatoid arthritis uye psoriasis.Izvi zvinobva zvaratidza anti-kuzvimba zvivakwa nekugadzirisa nzira dzakanangana nemhinduro yekuzvimba.Izvi zvinoratidza kukwanisa kwavo sevashandi vekurapa kwekugadzirisa zvirwere zvisingaperi uye zvirwere zvinosanganiswa.Uyezve, chikwata ichi chakaratidza basa mukati mehutano hwehutano (CNS).Yakaongororwa nekuda kwekugona kwayo muhutano hwetsinga hwakadai sechirwere cheAlzheimer uye chirwere cheParkinson.Iyo kompani inogona kuenzanisa ma receptors uye ma enzymes anosanganisirwa mukufambira mberi kwechirwere, achigona kupa neuroprotective mhedzisiro.Zvisinei, kumwe kutsvakurudza kunodiwa kuti unzwisise zvizere maitiro ayo ekuita uye kuongorora kushanda kwayo mukurapa zvirwere izvi zvakaoma. yl)phenyl] -4,5,6,7-tetrahydro-1H-pyrazolo[3,4-c]pyridine-3-carboxylic acid ethyl ester ine chivimbiso munzvimbo dzakawanda dzokurapa, kusanganisira anti-cancer, antibacterial, anti-inflammatory. , uye CNS kusagadzikana.Kugona kwayo kuri mukukwanisa kwayo kunanga nzira dzakanangana uye mareceptor anobatanidzwa mumamiriro aya.Nekudaro, kumwe kutsvagisa nekuferefeta kwakakosha kuti uongorore zvizere kugona kwayo, kukwidziridza zvimiro zvayo, uye kuongorora kuchengetedzeka kwayo uye kushanda kwayo muzvirongwa zvekiriniki.